α
1
Agonists
Antagonists
Abanoquil
Ajmalicine
Alfuzosin
Anisodamine
Anisodine
Atiprosin
Atypical antipsychotics
(e.g.,
brexpiprazole
,
clozapine
,
olanzapine
,
quetiapine
,
risperidone
)
Benoxathian
Beta blockers
(e.g.,
adimolol
,
amosulalol
,
arotinolol
,
carvedilol
,
eugenodilol
,
labetalol
)
Buflomedil
Bunazosin
Corynanthine
Dapiprazole
Domesticine
Doxazosin
Ergolines
(e.g.,
acetergamine
,
ergotamine
,
dihydroergotamine
,
lisuride
,
nicergoline
,
terguride
)
Etoperidone
Fenspiride
Hydroxyzine
Indoramin
Ketanserin
L-765,314
mCPP
Mepiprazole
Metazosin
Monatepil
Moxisylyte
Naftopidil
Nantenine
Neldazosin
Niaprazine
Niguldipine
Pardoprunox
Pelanserin
Perlapine
Phendioxan
Phenoxybenzamine
Phentolamine
Phenylpiperazine
antidepressants
(e.g.,
hydroxynefazodone
,
nefazodone
,
trazodone
,
triazoledione
)
Piperoxan
Prazosin
Quinazosin
Quinidine
Silodosin
Spegatrine
Spiperone
Talipexole
Tamsulosin
Terazosin
Tiodazosin
Tolazoline
Tetracyclic antidepressants
(e.g.,
amoxapine
,
maprotiline
,
mianserin
)
Tricyclic antidepressants
(e.g.,
amitriptyline
,
clomipramine
,
doxepin
,
imipramine
,
trimipramine
)
Trimazosin
Typical antipsychotics
(e.g.,
chlorpromazine
,
fluphenazine
,
loxapine
,
thioridazine
)
Urapidil
WB-4101
Zolertine
α
2
Agonists
Antagonists
1-PP
Adimolol
Amesergide
Aptazapine
Atipamezole
Atypical antipsychotics
(e.g.,
asenapine
,
brexpiprazole
,
clozapine
,
lurasidone
,
olanzapine
,
paliperidone
,
quetiapine
,
risperidone
,
zotepine
)
Azapirones
(e.g.,
buspirone
,
gepirone
,
ipsapirone
,
tandospirone
)
BRL-44408
Buflomedil
Cirazoline
Efaroxan
Esmirtazapine
Fenmetozole
Fluparoxan
Idazoxan
Ketanserin
Lisuride
mCPP
Mianserin
Mirtazapine
NAN-190
Pardoprunox
Phentolamine
Phenoxybenzamine
Piperoxan
Piribedil
Rauwolscine
Rotigotine
Setiptiline
Spegatrine
Spiroxatrine
Sunepitron
Terguride
Tolazoline
Typical antipsychotics
(e.g.,
chlorpromazine
,
fluphenazine
,
loxapine
,
thioridazine
)
Yohimbine
β
5-HT
1
5-HT
1A
Agonists:
8-OH-DPAT
Adatanserin
Amphetamine
Antidepressants
(e.g.,
etoperidone
,
hydroxynefazodone
,
nefazodone
,
trazodone
,
triazoledione
,
vilazodone
,
vortioxetine
)
Atypical antipsychotics
(e.g.,
aripiprazole
,
asenapine
,
brexpiprazole
,
cariprazine
,
clozapine
,
lurasidone
,
quetiapine
,
ziprasidone
)
Azapirones
(e.g.,
buspirone
,
eptapirone
,
gepirone
,
perospirone
,
tandospirone
)
Bay R 1531
Befiradol
BMY-14802
Cannabidiol
Dimemebfe
Dopamine
Ebalzotan
Eltoprazine
Enciprazine
Ergolines
(e.g.,
bromocriptine
,
cabergoline
,
dihydroergotamine
,
ergotamine
,
lisuride
,
LSD
,
methylergometrine (methylergonovine)
,
methysergide
,
pergolide
)
F-11,461
F-12826
F-13714
F-14679
F-15063
F-15,599
Flesinoxan
Flibanserin
Flumexadol
Hypidone
Lesopitron
LY-293284
LY-301317
mCPP
MKC-242
Naluzotan
NBUMP
Osemozotan
Oxaflozane
Pardoprunox
Piclozotan
Rauwolscine
Repinotan
Roxindole
RU-24,969
S-14,506
S-14671
S-15535
Sarizotan
Serotonin (5-HT)
SSR-181507
Sunepitron
Tryptamines
(e.g.,
5-CT
,
5-MeO-DMT
,
5-MT
,
bufotenin
,
DMT
,
indorenate
,
N-Me-5-HT
,
psilocin
,
psilocybin
)
TGBA01AD
U-92,016-A
Urapidil
Vilazodone
Xaliproden
Yohimbine
Antagonists:
Atypical antipsychotics
(e.g.,
iloperidone
,
risperidone
,
sertindole
)
AV965
Beta blockers
(e.g.,
alprenolol
,
carteolol
,
cyanopindolol
,
iodocyanopindolol
,
isamoltane
,
oxprenolol
,
penbutolol
,
pindobind
,
pindolol
,
propranolol
,
tertatolol
)
BMY-7,378
CSP-2503
Dotarizine
Ergolines
(e.g.,
metergoline
)
FCE-24379
Flopropione
GR-46611
Isamoltane
Lecozotan
Mefway
Metitepine (methiothepin)
MIN-117 (WF-516)
MPPF
NAN-190
Robalzotan
S-15535
SB-649,915
SDZ 216-525
Spiperone
Spiramide
Spiroxatrine
UH-301
WAY-100135
WAY-100635
Xylamidine
5-HT
1B
Agonists:
Anpirtoline
CGS-12066A
CP-93129
CP-94253
CP-122,288
CP-135807
Eltoprazine
Ergolines
(e.g.,
bromocriptine
,
dihydroergotamine
,
ergotamine
,
methylergometrine (methylergonovine)
,
methysergide
,
pergolide
)
mCPP
RU-24,969
Serotonin (5-HT)
Triptans
(e.g.,
avitriptan
,
donitriptan
,
eletriptan
,
sumatriptan
,
zolmitriptan
)
TFMPP
Tryptamines
(e.g.,
5-BT
,
5-CT
,
5-MT
,
DMT
)
Vortioxetine
5-HT
1D
Agonists:
CP-122,288
CP-135807
CP-286601
Ergolines
(e.g.,
bromocriptine
,
cabergoline
,
dihydroergotamine
,
ergotamine
,
LSD
,
methysergide
)
GR-46611
L-694247
L-772405
mCPP
PNU-109291
PNU-142633
Serotonin (5-HT)
TGBA01AD
Triptans
(e.g.,
almotriptan
,
avitriptan
,
donitriptan
,
eletriptan
,
frovatriptan
,
naratriptan
,
rizatriptan
,
sumatriptan
,
zolmitriptan
)
Tryptamines
(e.g.,
5-BT
,
5-CT
,
5-Et-DMT
,
5-MT
,
5-(nonyloxy)tryptamine
,
DMT
)
5-HT
1E
5-HT
1F
5-HT
2
5-HT
2A
Agonists:
25H/NB series (e.g.,
25I-NBF
,
25I-NBMD
,
25I-NBOH
,
25I-NBOMe
,
25B-NBOMe
,
25C-NBOMe
,
25TFM-NBOMe
,
2CBCB-NBOMe
,
25CN-NBOH
,
2CBFly-NBOMe
)
2Cs
(e.g.,
2C-B
,
2C-E
,
2C-I
,
2C-T-2
,
2C-T-7
,
2C-T-21
)
2C-B-FLY
2CB-Ind
5-Methoxytryptamines
(
5-MeO-DET
,
5-MeO-DiPT
,
5-MeO-DMT
,
5-MeO-DPT
,
5-MT
)
α-Alkyltryptamines
(e.g.,
5-Cl-αMT
,
5-Fl-αMT
,
5-MeO-αET
,
5-MeO-αMT
,
α-Me-5-HT
,
αET
,
αMT
)
AL-34662
AL-37350A
Bromo-DragonFLY
Dimemebfe
DMBMPP
DOx
(e.g.,
DOB
,
DOC
,
DOI
,
DOM
)
Efavirenz
Ergolines
(e.g.,
1P-LSD
,
ALD-52
,
bromocriptine
,
cabergoline
,
ergine (LSA)
,
ergometrine (ergonovine)
,
ergotamine
,
lisuride
,
LA-SS-Az
,
LSB
,
LSD
,
LSD-Pip
,
LSH
,
LSP
,
methylergometrine (methylergonovine)
,
pergolide
)
Flumexadol
IHCH-7113
Jimscaline
Lorcaserin
MDxx
(e.g.,
MDA (tenamfetamine)
,
MDMA (midomafetamine)
,
MDOH
,
MMDA
)
O-4310
Oxaflozane
PHA-57378
PNU-22394
PNU-181731
RH-34
SCHEMBL5334361
Phenethylamines
(e.g.,
lophophine
,
mescaline
)
Piperazines
(e.g.,
BZP
,
quipazine
,
TFMPP
)
Serotonin (5-HT)
TCB-2
TFMFly
Tryptamines
(e.g.,
5-BT
,
5-CT
,
bufotenin
,
DET
,
DiPT
,
DMT
,
DPT
,
psilocin
,
psilocybin
,
tryptamine
)
Antagonists:
5-I-R91150
5-MeO-NBpBrT
AC-90179
Adatanserin
Altanserin
Antihistamines
(e.g.,
cyproheptadine
,
hydroxyzine
,
ketotifen
,
perlapine
)
AMDA
Atypical antipsychotics
(e.g.,
amperozide
,
aripiprazole
,
asenapine
,
blonanserin
,
brexpiprazole
,
carpipramine
,
clocapramine
,
clorotepine
,
clozapine
,
fluperlapine
,
gevotroline
,
iloperidone
,
lurasidone
,
melperone
,
mosapramine
,
ocaperidone
,
olanzapine
,
paliperidone
,
quetiapine
,
risperidone
,
sertindole
,
zicronapine
,
ziprasidone
,
zotepine
)
Chlorprothixene
Cinanserin
CSP-2503
Deramciclane
Dotarizine
Eplivanserin
Ergolines
(e.g.,
amesergide
,
LY-53857
,
LY-215,840
,
mesulergine
,
metergoline
,
methysergide
,
sergolexole
)
Fananserin
Flibanserin
Glemanserin
Irindalone
Ketanserin
KML-010
Landipirdine
LY-393558
mCPP
Medifoxamine
Metitepine (methiothepin)
MIN-117 (WF-516)
Naftidrofuryl
Nantenine
Nelotanserin
Opiranserin (VVZ-149)
Pelanserin
Phenoxybenzamine
Pimavanserin
Pirenperone
Pizotifen
Pruvanserin
Rauwolscine
Ritanserin
Roluperidone
S-14671
Sarpogrelate
Serotonin antagonists and reuptake inhibitors
(e.g.,
etoperidone
,
hydroxynefazodone
,
lubazodone
,
mepiprazole
,
nefazodone
,
triazoledione
,
trazodone
)
SR-46349B
TGBA01AD
Teniloxazine
Temanogrel
Tetracyclic antidepressants
(e.g.,
amoxapine
,
aptazapine
,
esmirtazapine
,
maprotiline
,
mianserin
,
mirtazapine
)
Tricyclic antidepressants
(e.g.,
amitriptyline
)
Typical antipsychotics
(e.g.,
chlorpromazine
,
fluphenazine
,
haloperidol
,
loxapine
,
perphenazine
,
pimozide
,
pipamperone
,
prochlorperazine
,
setoperone
,
spiperone
,
spiramide
,
thioridazine
,
thiothixene
,
trifluoperazine
)
Volinanserin
Xylamidine
Yohimbine
5-HT
2B
Agonists:
4-Methylaminorex
Aminorex
Amphetamines
(e.g.,
chlorphentermine
,
cloforex
,
dexfenfluramine
,
fenfluramine
,
levofenfluramine
,
norfenfluramine
)
BW-723C86
DOx
(e.g.,
DOB
,
DOC
,
DOI
,
DOM
)
Ergolines
(e.g.,
cabergoline
,
dihydroergocryptine
,
dihydroergotamine
,
ergotamine
,
methylergometrine (methylergonovine)
,
methysergide
,
pergolide
)
Lorcaserin
MDxx
(e.g.,
MDA (tenamfetamine)
,
MDMA (midomafetamine)
,
MDOH
,
MMDA
)
Piperazines
(e.g.,
TFMPP
)
PNU-22394
Ro60-0175
Serotonin (5-HT)
Tryptamines
(e.g.,
5-BT
,
5-CT
,
5-MT
,
α-Me-5-HT
,
bufotenin
,
DET
,
DiPT
,
DMT
,
DPT
,
psilocin
,
psilocybin
,
tryptamine
)
Antagonists:
Agomelatine
Atypical antipsychotics
(e.g.,
amisulpride
,
aripiprazole
,
asenapine
,
brexpiprazole
,
cariprazine
,
clozapine
,
N-desalkylquetiapine (norquetiapine)
,
N-desmethylclozapine (norclozapine)
,
olanzapine
,
pipamperone
,
quetiapine
,
risperidone
,
ziprasidone
)
Cyproheptadine
EGIS-7625
Ergolines
(e.g.,
amesergide
,
bromocriptine
,
lisuride
,
LY-53857
,
LY-272015
,
mesulergine
)
Ketanserin
LY-393558
mCPP
Metadoxine
Metitepine (methiothepin)
Pirenperone
Pizotifen
Propranolol
PRX-08066
Rauwolscine
Ritanserin
RS-127445
Sarpogrelate
SB-200646
SB-204741
SB-206553
SB-215505
SB-221284
SB-228357
SDZ SER-082
Tegaserod
Tetracyclic antidepressants
(e.g.,
amoxapine
,
mianserin
,
mirtazapine
)
Trazodone
Typical antipsychotics
(e.g.,
chlorpromazine
)
TIK-301
Yohimbine
5-HT
2C
Agonists:
2Cs
(e.g.,
2C-B
,
2C-E
,
2C-I
,
2C-T-2
,
2C-T-7
,
2C-T-21
)
5-Methoxytryptamines
(
5-MeO-DET
,
5-MeO-DiPT
,
5-MeO-DMT
,
5-MeO-DPT
,
5-MT
)
α-Alkyltryptamines
(e.g.,
5-Cl-αMT
,
5-Fl-αMT
,
5-MeO-αET
,
5-MeO-αMT
,
α-Me-5-HT
,
αET
,
αMT
)
A-372159
AL-38022A
Alstonine
CP-809101
Dimemebfe
DOx
(e.g.,
DOB
,
DOC
,
DOI
,
DOM
)
Ergolines
(e.g.,
ALD-52
,
cabergoline
,
dihydroergotamine
,
ergine (LSA)
,
ergotamine
,
lisuride
,
LA-SS-Az
,
LSB
,
LSD
,
LSD-Pip
,
LSH
,
LSP
,
pergolide
)
Flumexadol
Lorcaserin
MDxx
(e.g.,
MDA (tenamfetamine)
,
MDMA (midomafetamine)
,
MDOH
,
MMDA
)
MK-212
ORG-12962
ORG-37684
Oxaflozane
PHA-57378
Phenethylamines
(e.g.,
lophophine
,
mescaline
)
Piperazines
(e.g.,
aripiprazole
,
BZP
,
mCPP
,
quipazine
,
TFMPP
)
PNU-22394
PNU-181731
Ro60-0175
Ro60-0213
Serotonin (5-HT)
Tryptamines
(e.g.,
5-BT
,
5-CT
,
bufotenin
,
DET
,
DiPT
,
DMT
,
DPT
,
psilocin
,
psilocybin
,
tryptamine
)
Vabicaserin
WAY-629
WAY-161503
YM-348
Antagonists:
Adatanserin
Agomelatine
Atypical antipsychotics
(e.g.,
asenapine
,
clorotepine
,
clozapine
,
fluperlapine
,
iloperidone
,
melperone
,
olanzapine
,
paliperidone
,
quetiapine
,
risperidone
,
sertindole
,
ziprasidone
,
zotepine
)
Captodiame
CEPC
Cinanserin
Cyproheptadine
Deramciclane
Desmetramadol
Dotarizine
Eltoprazine
Ergolines
(e.g.,
amesergide
,
bromocriptine
,
LY-53857
,
LY-215,840
,
mesulergine
,
metergoline
,
methysergide
,
sergolexole
)
Etoperidone
Fluoxetine
FR-260010
Irindalone
Ketanserin
Ketotifen
Latrepirdine (dimebolin)
Medifoxamine
Metitepine (methiothepin)
Nefazodone
Pirenperone
Pizotifen
Propranolol
Ritanserin
RS-102221
S-14671
SB-200646
SB-206553
SB-221284
SB-228357
SB-242084
SB-243213
SDZ SER-082
Tedatioxetine
Tetracyclic antidepressants
(e.g.,
amoxapine
,
aptazapine
,
esmirtazapine
,
maprotiline
,
mianserin
,
mirtazapine
)
TIK-301
Tramadol
Trazodone
Tricyclic antidepressants
(e.g.,
amitriptyline
,
nortriptyline
)
Typical antipsychotics
(e.g.,
chlorpromazine
,
loxapine
,
pimozide
,
pipamperone
,
thioridazine
)
Xylamidine
5-HT
3
–
7
5-HT
3
Agonists:
Alcohols
(e.g.,
butanol
,
ethanol (alcohol)
,
trichloroethanol
)
m-CPBG
Phenylbiguanide
Piperazines
(e.g.,
BZP
,
mCPP
,
quipazine
)
RS-56812
Serotonin (5-HT)
SR-57227
SR-57227A
Tryptamines
(e.g.,
2-Me-5-HT
,
5-CT
,
bufotenidine (5-HTQ)
)
Volatiles/gases
(e.g.,
halothane
,
isoflurane
,
toluene
,
trichloroethane
)
YM-31636
Antagonists:
Alosetron
Anpirtoline
Arazasetron
AS-8112
Atypical antipsychotics
(e.g.,
clozapine
,
olanzapine
,
quetiapine
)
Azasetron
Batanopride
Bemesetron (MDL-72222)
Bupropion
Cilansetron
CSP-2503
Dazopride
Dolasetron
Galanolactone
Granisetron
Hydroxybupropion
Lerisetron
Memantine
Ondansetron
Palonosetron
Ramosetron
Renzapride
Ricasetron
Tedatioxetine
Tetracyclic antidepressants
(e.g.,
amoxapine
,
mianserin
,
mirtazapine
)
Thujone
Tropanserin
Tropisetron
Typical antipsychotics
(e.g.,
loxapine
)
Volatiles/gases
(e.g.,
nitrous oxide
,
sevoflurane
,
xenon
)
Vortioxetine
Zacopride
Zatosetron
5-HT
4
5-HT
5A
5-HT
6
Agonists:
Ergolines
(e.g.,
dihydroergocryptine
,
dihydroergotamine
,
ergotamine
,
lisuride
,
LSD
,
mesulergine
,
metergoline
,
methysergide
)
Hypidone
Serotonin (5-HT)
Tryptamines
(e.g.,
2-Me-5-HT
,
5-BT
,
5-CT
,
5-MT
,
Bufotenin
,
E-6801
,
E-6837
,
EMD-386088
,
EMDT
,
LY-586713
,
N-Me-5-HT
,
ST-1936
,
tryptamine
)
WAY-181187
WAY-208466
Antagonists:
ABT-354
Atypical antipsychotics
(e.g.,
aripiprazole
,
asenapine
,
clorotepine
,
clozapine
,
fluperlapine
,
iloperidone
,
olanzapine
,
tiospirone
)
AVN-101
AVN-211
AVN-322
AVN-397
BGC20-760
BVT-5182
BVT-74316
Cerlapirdine
EGIS-12,233
GW-742457
Idalopirdine
Ketanserin
Landipirdine
Latrepirdine (dimebolin)
Masupirdine
Metitepine (methiothepin)
MS-245
PRX-07034
Ritanserin
Ro 04-6790
Ro 63-0563
SB-258585
SB-271046
SB-357134
SB-399885
SB-742457
Tetracyclic antidepressants
(e.g.,
amoxapine
,
mianserin
)
Tricyclic antidepressants
(e.g.,
amitriptyline
,
clomipramine
,
doxepin
,
nortriptyline
)
Typical antipsychotics
(e.g.,
chlorpromazine
,
loxapine
)
5-HT
7
Antagonists:
Atypical antipsychotics
(e.g.,
amisulpride
,
aripiprazole
,
asenapine
,
brexpiprazole
,
clorotepine
,
clozapine
,
fluperlapine
,
olanzapine
,
risperidone
,
sertindole
,
tiospirone
,
ziprasidone
,
zotepine
)
Butaclamol
DR-4485
EGIS-12,233
Ergolines
(e.g.,
2-Br-LSD (BOL-148)
,
amesergide
,
bromocriptine
,
cabergoline
,
dihydroergotamine
,
ergotamine
,
LY-53857
,
LY-215,840
,
mesulergine
,
metergoline
,
methysergide
,
sergolexole
)
JNJ-18038683
Ketanserin
LY-215,840
Metitepine (methiothepin)
Ritanserin
SB-258719
SB-258741
SB-269970
SB-656104
SB-656104A
SB-691673
SLV-313
SLV-314
Spiperone
SSR-181507
Tetracyclic antidepressants
(e.g.,
amoxapine
,
maprotiline
,
mianserin
,
mirtazapine
)
Tricyclic antidepressants
(e.g.,
amitriptyline
,
clomipramine
,
imipramine
)
Typical antipsychotics
(e.g.,
acetophenazine
,
chlorpromazine
,
chlorprothixene
,
fluphenazine
,
loxapine
,
pimozide
)
Vortioxetine